Antibody-Drug Conjugate (ADC)Population PK (2-CMT ADC + 1-CMT DM4 Payload)IV InfusionOncology / Ovarian Cancer

Mirvetuximab Soravtansine (ELAHERE) PopPK

Indication: FRα-positive, platinum-resistant epithelial ovarian, fallopian tube, or primary peritoneal cancer; maytansinoid DM4 payload

Population PK simulator for mirvetuximab soravtansine (ELAHERE, IMGN853) — FRα-targeted ADC with DM4 maytansinoid payload for platinum-resistant ovarian cancer. Two-compartment ADC model with albumin covariate on clearance and AIBW-based dosing. The first ADC to show OS benefit vs chemotherapy in a solid tumor (MIRASOL trial). Based on Choudhry et al. CPT 2023 and FDA Clinical Pharmacology Review.

Drug Overview

Clinical Context

Molecular Target
FRα (Folate Receptor Alpha, FOLR1)
Drug Class
Antibody-Drug Conjugate (ADC)
Therapeutic Area
Oncology / Ovarian Cancer
Indication
FRα-positive, platinum-resistant epithelial ovarian, fallopian tube, or primary peritoneal cancer; maytansinoid DM4 payload
Route of Administration
IV Infusion

Model Information

Model Type
Population PK (2-CMT ADC + 1-CMT DM4 Payload)

This simulator was built from published pharmacometric literature using PKPDBuilder's AI-powered model extraction pipeline.

Pharmacokinetic Parameters

Additional Parameters

ParameterValue
k120.22
k210.3
ADC CL0.65
DM4 Vd420
Standard Dose6
DM4 Payload CL38
ADC V1 (Central)3.8
ADC V2 (Peripheral)2.1
Albumin Exponent on CL0.45
Payload Release Rate (kr)0.008

Parameters sourced from published population pharmacokinetic models. Values represent typical population estimates; individual patient parameters may vary.

About This Simulator

This interactive pharmacokinetic simulator for Mirvetuximab Soravtansine (ELAHERE) allows you to explore concentration-time profiles under different dosing scenarios. The underlying Population PK (2-CMT ADC + 1-CMT DM4 Payload) model characterizes the pharmacokinetics of this antibody-drug conjugate (adc) following iv infusion administration.

Use the simulator to visualize key exposure metrics including AUC (area under the curve), Cmax (peak concentration), and Ctrough (trough concentration).

Built with PKPDBuilder — an AI-powered platform that transforms published pharmacometric literature into interactive, deployable Shiny applications. No coding required.

Frequently Asked Questions

What is the Mirvetuximab Soravtansine (ELAHERE) PK simulator?

This is a free, interactive pharmacokinetic simulator for Mirvetuximab Soravtansine (ELAHERE) used in FRα-positive, platinum-resistant epithelial ovarian, fallopian tube, or primary peritoneal cancer; maytansinoid DM4 payload. It allows researchers, pharmacologists, and students to explore concentration-time profiles, dosing regimens, and exposure metrics based on published population PK models.

What drug class does Mirvetuximab Soravtansine (ELAHERE) belong to?

Mirvetuximab Soravtansine (ELAHERE) is classified as a Antibody-Drug Conjugate (ADC) that targets FRα (Folate Receptor Alpha, FOLR1). It is used in the Oncology / Ovarian Cancer therapeutic area.

What route of administration does this model simulate?

This simulator models IV Infusion administration of Mirvetuximab Soravtansine (ELAHERE). The pharmacokinetic parameters (absorption rate, bioavailability, volume of distribution) are specific to this route.

What type of PK model is used?

This simulator uses a Population PK (2-CMT ADC + 1-CMT DM4 Payload) model. This model characterizes the time-course of drug concentrations following dosing.

Is this simulator free to use?

Yes, all PKPDBuilder simulators are completely free. They are built from published pharmacokinetic literature and are intended for research and educational purposes. No login is required to run simulations.

Can I use this for clinical dosing decisions?

No. This simulator is for research and educational purposes only. It should not be used for clinical decision-making or patient dosing. Always consult the prescribing information and clinical pharmacology guidelines for therapeutic drug use.

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⚠️ Disclaimer

This simulator is for research and educational purposes only. It is not intended for clinical decision-making, patient dosing, or therapeutic drug monitoring. Pharmacokinetic parameters are derived from published literature and represent population-level estimates. Individual patient pharmacokinetics may differ significantly. Always consult approved prescribing information and qualified healthcare professionals for clinical decisions.

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