Pharmacokinetics Guides
Comprehensive PK parameter guides for 181+ drugs. Each guide includes key pharmacokinetic data, dosing information, and an interactive simulator.
5-Fluorouracil Pharmacokinetics Guide
Cancer chemotherapy
Antimetabolite
Read guide →ADC Effector Function Model Pharmacokinetics Guide
Solid Tumors
ADC
Read guide →ADCs Pharmacokinetics Guide
HER2-positive breast cancer, NSCLC, gastric/GEJ cancer
Antibody-Drug Conjugate (ADC)
Read guide →Abc Pharmacokinetics Guide
Benign prostatic hyperplasia (BPH), hypertension
Alpha-1 Adrenoceptor Antagonist
Read guide →Acetaminophen Pharmacokinetics Guide
Pain/Fever
Analgesic
Read guide →Amikacine Pharmacokinetics Guide
Severe infections in ICU patients including sepsis and nosocomial pneumonia
Aminoglycoside antibiotic
Read guide →Amlitelimab Pharmacokinetics Guide
Atopic Dermatitis
mAb
Read guide →Antibiotic PD Interaction Pharmacokinetics Guide
Bacterial infections
Antibiotics
Read guide →Asundexian FXIa Inhibitor Pharmacokinetics Guide
Anticoagulation
Small Molecule
Read guide →BTK Degrader Pharmacokinetics Guide
B-cell Malignancies
PROTAC
Read guide →BTK Targeted Degrader Pharmacokinetics Guide
B-cell Malignancies
PROTAC
Read guide →Bedaquiline trial Pharmacokinetics Guide
Multi-drug resistant tuberculosis (MDR-TB)
Diarylquinoline antimycobacterial
Read guide →Betamethasone Metabolite Pharmacokinetics Guide
Inflammation/Preterm Labor
Small Molecule
Read guide →Betamethasone NCA Pharmacokinetics Guide
Inflammation
Small Molecule
Read guide →Biktarvy (Bictegravir/Emtricitabine/TAF) Pharmacokinetics Guide
HIV-1 infection
Small Molecule
Read guide →Carbamazepine TDM Pharmacokinetics Guide
Epilepsy
Anticonvulsant
Read guide →Cefepime "Jonckheere" Pharmacokinetics Guide
Nosocomial infections, febrile neutropenia, severe bacterial infections in ICU
Beta-Lactam Antibiotic (4th-gen Cephalosporin)
Read guide →Ciprofloxacin Pharmacokinetics Guide
Bacterial infections
Fluoroquinolone
Read guide →Cisplatin Pharmacokinetics Guide
Cancer chemotherapy
Platinum
Read guide →Concizumab Pharmacokinetics Guide
Hemophilia
mAb
Read guide →Cosentyx (Secukinumab) Pharmacokinetics Guide
Plaque psoriasis
mAb
Read guide →Cyclosporine Pharmacokinetics Guide
Organ Transplant Rejection
Small Molecule
Read guide →Cyclosporine TDM Pharmacokinetics Guide
Transplant immunosuppression
Calcineurin inhibitor
Read guide →DAC Pharmacokinetics Guide
Multiple Sclerosis
Monoclonal Antibody (Anti-CD25)
Read guide →DTg Pharmacokinetics Guide
HIV-1 infection (antiretroviral therapy)
Integrase Strand Transfer Inhibitor (INSTI)
Read guide →Darzalex (Daratumumab) Pharmacokinetics Guide
Multiple myeloma
mAb
Read guide →Dato Pharmacokinetics Guide
TROP2-positive metastatic breast cancer
Antibody-Drug Conjugate (ADC)
Read guide →Datroway Pharmacokinetics Guide
Locally advanced or metastatic non-squamous NSCLC (TROPION-Lung08), HR+/HER2-low/negative metastatic breast cancer (TROPION-Breast01), and triple-negative breast cancer; TROP2-directed ADC with DXd payload
Antibody-Drug Conjugate (ADC)
Read guide →Digoxin Pharmacokinetics Guide
Heart Failure / Atrial Fibrillation
Small Molecule
Read guide →Digoxin TDM Pharmacokinetics Guide
Heart failure/AF
Cardiac glycoside
Read guide →Donidalorsen Pharmacokinetics Guide
Hereditary Angioedema
ASO
Read guide →Doxorubicin Pharmacokinetics Guide
Cancer chemotherapy
Anthracycline
Read guide →Dupilumab Pharmacokinetics Guide
Atopic Dermatitis
mAb
Read guide →Dupilumab Population Pharmacokinetics Guide
Atopic Dermatitis
mAb
Read guide →Dupixent (Dupilumab) Pharmacokinetics Guide
Atopic dermatitis
mAb
Read guide →Efsubaglutide Alfa Pharmacokinetics Guide
Type 2 Diabetes
GLP-1 Receptor Agonist
Read guide →Eliquis (Apixaban) Pharmacokinetics Guide
Stroke prevention in atrial fibrillation
Small Molecule
Read guide →Empagliflozin Pharmacokinetics Guide
Type 2 Diabetes Mellitus
SGLT2 inhibitor
Read guide →Enbrel (Etanercept) Pharmacokinetics Guide
Rheumatoid arthritis
Fusion Protein
Read guide →Enhertu Pharmacokinetics Guide
HER2-positive breast cancer, gastric/gastroesophageal adenocarcinoma, NSCLC
Antibody-Drug Conjugate (ADC)
Read guide →Entresto (Sacubitril/Valsartan) Pharmacokinetics Guide
Heart failure with reduced ejection fraction
Small Molecule
Read guide →Entyvio (Vedolizumab) Pharmacokinetics Guide
Ulcerative colitis
mAb
Read guide →Eplontersen Pharmacokinetics Guide
Hereditary transthyretin-mediated amyloidosis (hATTR)
Antisense Oligonucleotide (ASO)
Read guide →Eylea (Aflibercept) Pharmacokinetics Guide
Wet age-related macular degeneration
Fusion Protein
Read guide →Farxiga (Dapagliflozin) Pharmacokinetics Guide
Type 2 diabetes mellitus
Small Molecule
Read guide →Flutamide PBPK Model Pharmacokinetics Guide
Stage D2 metastatic prostate cancer (combined with LHRH agonist)
Non-steroidal Antiandrogen
Read guide →Fruquintinib Pharmacokinetics Guide
Metastatic Colorectal Cancer
VEGFR Tyrosine Kinase Inhibitor
Read guide →Ganciclovir Pharmacokinetics Guide
CMV Infection
Small Molecule
Read guide →Gentamicin TDM Pharmacokinetics Guide
Bacterial infections
Aminoglycoside
Read guide →Givosiran ALA Pharmacokinetics Guide
Acute Hepatic Porphyria
siRNA
Read guide →Givosiran Pharmacokinetics Guide
Acute Hepatic Porphyria
siRNA
Read guide →Hemlibra (Emicizumab) Pharmacokinetics Guide
Hemophilia A
Bispecific mAb
Read guide →Humira (Adalimumab) Pharmacokinetics Guide
Rheumatoid arthritis
mAb
Read guide →Ibrance (Palbociclib) Pharmacokinetics Guide
HR+/HER2- metastatic breast cancer
Small Molecule
Read guide →Imatinib Pharmacokinetics Guide
CML / GIST
Small Molecule
Read guide →Imbruvica (Ibrutinib) Pharmacokinetics Guide
Chronic lymphocytic leukemia
Small Molecule
Read guide →Imfinzi (Durvalumab) Pharmacokinetics Guide
Non-small cell lung cancer
mAb
Read guide →Implémentation modèle Vezina Pharmacokinetics Guide
Antiviral — Nucleoside Analogue
Read guide →Infigratinib Pharmacokinetics Guide
Cholangiocarcinoma
Small Molecule
Read guide →Inotersen Pharmacokinetics Guide
Hereditary transthyretin-mediated amyloidosis polyneuropathy (hATTR-PN)
Antisense Oligonucleotide (ASO)
Read guide →Insulin Pharmacokinetics Guide
DKA/Diabetes
Hormone
Read guide →Invega Sustenna (Paliperidone Palmitate) Pharmacokinetics Guide
Schizophrenia
Small Molecule
Read guide →Jardiance (Empagliflozin) Pharmacokinetics Guide
Type 2 diabetes mellitus
Small Molecule
Read guide →Keytruda (Pembrolizumab) Pharmacokinetics Guide
Melanoma and non-small cell lung cancer
mAb
Read guide →Keytruda Pharmacokinetics Guide
Cancer immunotherapy
PD-1 inhibitor
Read guide →Kovaltry Pharmacokinetics Guide
Hemophilia A prophylaxis and treatment
Recombinant Factor VIII (Antihemophilic Factor)
Read guide →Lynparza (Olaparib) Pharmacokinetics Guide
BRCA-mutated ovarian cancer
Small Molecule
Read guide →MTXPK Pharmacokinetics Guide
Acute lymphoblastic leukemia (ALL), osteosarcoma
Antifolate antineoplastic
Read guide →Maternal-Fetal Pharmacokinetics Guide
Maternal-Fetal Medicine
Small Molecule
Read guide →Methotrexate High-Dose Pharmacokinetics Guide
Cancer/RA
Antimetabolite
Read guide →Midazolam Pharmacokinetics Guide
Sedation
Benzodiazepine
Read guide →Minimal Antibody PBPK Pharmacokinetics Guide
Monoclonal Antibodies
mAb
Read guide →Mirvetuximab Soravtansine (ELAHERE) Pharmacokinetics Guide
FRα-positive, platinum-resistant epithelial ovarian, fallopian tube, or primary peritoneal cancer; maytansinoid DM4 payload
Antibody-Drug Conjugate (ADC)
Read guide →Modèle Caldes Pharmacokinetics Guide
Antiviral
Read guide →Modèle Chen Pharmacokinetics Guide
Antiviral
Read guide →Morphine Pharmacokinetics Guide
Pain management
Opioid
Read guide →Mounjaro (Tirzepatide) Pharmacokinetics Guide
Type 2 diabetes mellitus
Dual GIP/GLP-1 RA
Read guide →Moxifloxacin Pediatric Pharmacokinetics Guide
Pediatric Tuberculosis
Fluoroquinolone Antibiotic
Read guide →Mycophenolate Pharmacokinetics Guide
Organ Transplant Rejection
Small Molecule
Read guide →NCA BET Pharmacokinetics Guide
Antenatal corticosteroid therapy for fetal lung maturation; placental transfer characterization
Corticosteroid
Read guide →OXZ_PopPK Pharmacokinetics Guide
Partial-onset seizures in adults and children ≥ 2 years
Antiepileptic Drug (AED)
Read guide →Ocrevus (Ocrelizumab) Pharmacokinetics Guide
Multiple sclerosis
mAb
Read guide →Ofev (Nintedanib) Pharmacokinetics Guide
Idiopathic pulmonary fibrosis
Small Molecule
Read guide →Oncology Dose Selection Tool Pharmacokinetics Guide
Solid Tumors
Small Molecule
Read guide →Opdivo (Nivolumab) Pharmacokinetics Guide
Melanoma and non-small cell lung cancer
mAb
Read guide →Orencia (Abatacept) Pharmacokinetics Guide
Rheumatoid arthritis
Fusion Protein
Read guide →Oxacillin Neonatal Pharmacokinetics Guide
MSSA Infections (Neonates)
Small Molecule
Read guide →Oxfendazole Population Pharmacokinetics Guide
Onchocerciasis (river blindness)
Benzimidazole Anthelminthic
Read guide →Ozempic (Semaglutide) Pharmacokinetics Guide
Type 2 diabetes mellitus
GLP-1 RA
Read guide →PBPK-PD Topo1-Based ADC Pharmacokinetics Guide
Solid tumors (breast, lung, gastric, colorectal cancer)
Antibody-Drug Conjugate (ADC)
Read guide →PBPK-PD Topo1-Based ADC Pharmacokinetics Guide
Solid tumors (HER2-positive and Trop-2-positive cancers)
Antibody-Drug Conjugate
Read guide →PBPK-PD Topo1-Based ADC Pharmacokinetics Guide
Solid tumors (breast, lung, gastric, colorectal cancer)
Antibody-Drug Conjugate (ADC)
Read guide →PBPK-PD of ADCs Pharmacokinetics Guide
Antibody-Drug Conjugate (ADC)
Read guide →PKPD model for lesinurad (Zurampic) Pharmacokinetics Guide
Hyperuricemia associated with gout (combination with xanthine oxidase inhibitors)
Xanthine Oxidase Inhibitors / Uricosurics
Read guide →Paclitaxel Pharmacokinetics Guide
Cancer chemotherapy
Taxane
Read guide →Patritumab Deruxtecan (HER3-DXd) Pharmacokinetics Guide
EGFR-mutant NSCLC after EGFR TKI and platinum therapy; HER3-directed ADC with DXd payload
Antibody-Drug Conjugate (ADC)
Read guide →Paxlovid (Nirmatrelvir/Ritonavir) Pharmacokinetics Guide
COVID-19 treatment
Small Molecule
Read guide →Perjeta (Pertuzumab) Pharmacokinetics Guide
HER2-positive breast cancer
mAb
Read guide →Phenytoin TDM Pharmacokinetics Guide
Epilepsy
Anticonvulsant
Read guide →Piperacilin Pharmacokinetics Guide
Beta-lactam Antibiotic
Read guide →Pomalyst (Pomalidomide) Pharmacokinetics Guide
Multiple myeloma
Small Molecule
Read guide →Pop Pharmacokinetics Guide
Hypertension
Angiotensin II Receptor Blocker (ARB)
Read guide →PopPK Framework Model Pharmacokinetics Guide
Drug Development
Small Molecule
Read guide →PopPK of Docetaxel Pharmacokinetics Guide
Taxane (Microtubule Stabilizer)
Read guide →Population model of Linezolid in ARDS on vvECMO Pharmacokinetics Guide
Oxazolidinone antibiotic
Read guide →Pravastatin EHC Model Pharmacokinetics Guide
Hypercholesterolemia
Statin
Read guide →Pravastatin SLCO1B1 PGx Model Pharmacokinetics Guide
Hypercholesterolemia
Statin
Read guide →Prolia (Denosumab) Pharmacokinetics Guide
Postmenopausal osteoporosis
mAb
Read guide →QSP Platform Model Pharmacokinetics Guide
Drug Development
Platform
Read guide →RMC Pharmacokinetics Guide
ALK/ROS1 Inhibitor (2nd generation)
Read guide →Revlimid (Lenalidomide) Pharmacokinetics Guide
Multiple myeloma
Small Molecule
Read guide →Rifampicin Pharmacokinetics Guide
Tuberculosis
Rifamycin
Read guide →Rifapentine Pharmacokinetics Guide
Tuberculosis treatment and latent TB infection prophylaxis
Rifamycin antibiotic
Read guide →Rinvoq (Upadacitinib) Pharmacokinetics Guide
Rheumatoid arthritis
Small Molecule
Read guide →Risperidone D2RO Pharmacokinetics Guide
Schizophrenia
Small Molecule
Read guide →Ruc Pharmacokinetics Guide
BRCA-mutant and HRD+ breast cancer
PARP inhibitor
Read guide →Rybelsus (Oral Semaglutide) Pharmacokinetics Guide
Type 2 diabetes mellitus
GLP-1 RA
Read guide →Semaglutide Pharmacokinetics Guide
Type 2 Diabetes / Obesity
GLP-1 RA
Read guide →Sertraline Pharmacokinetics Guide
SSRI Antidepressant
Read guide →Simvastatin Pharmacokinetics Guide
Hypercholesterolemia
Statin
Read guide →Skyrizi (Risankizumab) Pharmacokinetics Guide
Plaque psoriasis
mAb
Read guide →Stelara (Ustekinumab) Pharmacokinetics Guide
Plaque psoriasis
mAb
Read guide →T-DXd (Enhertu) PBPK-PD ILD Risk Pharmacokinetics Guide
HER2-positive metastatic breast cancer, gastric/GEJ adenocarcinoma, NSCLC, and other HER2-expressing solid tumors; ILD risk stratification and dose optimization
Antibody-Drug Conjugate (ADC)
Read guide →T-cell Engager Pharmacokinetics Guide
Hematologic Malignancies
mAb
Read guide →TMDD Model Pharmacokinetics Guide
HER2-positive Breast Cancer
Monoclonal Antibody (Anti-HER2)
Read guide →TMDD Model 3 Pharmacokinetics Guide
Monoclonal Antibody (anti-HER2)
Read guide →TMDD Model 4 Pharmacokinetics Guide
Monoclonal Antibody (HER2-targeted)
Read guide →Tacro2 Pharmacokinetics Guide
Allogeneic hematopoietic cell transplantation (allo-HCT)
Calcineurin Inhibitor
Read guide →Tacrolimus Pharmacokinetics Guide
Organ Transplant
Small Molecule
Read guide →Tacrolimus TDM Pharmacokinetics Guide
Transplant immunosuppression
Calcineurin inhibitor
Read guide →Tacrolimus model Pharmacokinetics Guide
Kidney transplant immunosuppression
Calcineurin inhibitor (Immunosuppressant)
Read guide →Tacrolimus pop Pharmacokinetics Guide
Pediatric/young adult hematopoietic cell transplantation
Calcineurin inhibitor (immunosuppressant)
Read guide →Tagrisso (Osimertinib) Pharmacokinetics Guide
EGFR-mutated non-small cell lung cancer
Small Molecule
Read guide →Tapering- Venlafaxine Pharmacokinetics Guide
Major depressive disorder, generalized anxiety disorder — antidepressant tapering and withdrawal risk assessment
Antidepressants (SSRI, SNRI, NaSSA)
Read guide →Tecentriq (Atezolizumab) Pharmacokinetics Guide
Non-small cell lung cancer
mAb
Read guide →TehopyllineTest Pharmacokinetics Guide
Asthma, COPD, neonatal apnea
Methylxanthine bronchodilator
Read guide →Test Pharmacokinetics Guide
Opioid overdose reversal (synthetic opioid and fentanyl exposure)
Opioid Antagonists
Read guide →Test Pharmacokinetics Guide
Opioid overdose reversal (synthetic opioid and fentanyl exposure)
Opioid Receptor Antagonists
Read guide →Test Complete Pharmacokinetics Guide
Read guide →Theophylline TDM Pharmacokinetics Guide
Asthma/COPD
Methylxanthine
Read guide →Torsemide Pharmacokinetics Guide
Heart Failure, Edema
Loop Diuretic
Read guide →Tramadol Pharmacokinetics Guide
Neuropathic Pain
Opioid Analgesic
Read guide →Trastuzumab (Herceptin) PBPK-TMDD Pharmacokinetics Guide
HER2-positive breast cancer
Anti-HER2 Monoclonal Antibody
Read guide →Trastuzumab Pharmacokinetics Guide
HER2+ Breast Cancer
mAb
Read guide →Trastuzumab Pharmacokinetics Guide
HER2+ Breast Cancer
mAb
Read guide →Trastuzumab Pharmacokinetics Guide
Monoclonal Antibody
Read guide →Tremfya (Guselkumab) Pharmacokinetics Guide
Plaque psoriasis
mAb
Read guide →Trikafta (Elexacaftor/Tezacaftor/Ivacaftor) Pharmacokinetics Guide
Cystic fibrosis
Small Molecule
Read guide →Trodelvy Pharmacokinetics Guide
Unresectable locally advanced or metastatic triple-negative breast cancer (mTNBC), HR+/HER2-negative metastatic breast cancer after endocrine and CDK4/6 inhibitor therapy, and locally advanced or metastatic urothelial cancer; TROP2-directed ADC with SN-38 payload
Antibody-Drug Conjugate (ADC)
Read guide →Trulicity (Dulaglutide) Pharmacokinetics Guide
Type 2 diabetes mellitus
GLP-1 RA
Read guide →Tumor Exposure Analysis Model Pharmacokinetics Guide
Solid Tumors
mAb
Read guide →VRC07-523-LS Pharmacokinetics Guide
HIV prevention in infants and adults
Broadly Neutralizing Antibody (bNAb)
Read guide →Vabysmo (Faricimab) Pharmacokinetics Guide
Wet age-related macular degeneration
Bispecific mAb
Read guide →Vancomycin TDM Pharmacokinetics Guide
Bacterial infections
Glycopeptide
Read guide →Verzenio (Abemaciclib) Pharmacokinetics Guide
HR+/HER2- metastatic breast cancer
Small Molecule
Read guide →Voriconazole Pharmacokinetics Guide
Invasive aspergillosis, candidemia
Triazole Antifungal
Read guide →Voriconazole IV Pharmacokinetics Guide
Invasive Fungal Infections
Small Molecule
Read guide →Vortioxetine Pharmacokinetics Guide
Major Depressive Disorder (MDD)
Antidepressant (Multimodal)
Read guide →Vyndaqel (Tafamidis) Pharmacokinetics Guide
Transthyretin amyloid cardiomyopathy
Small Molecule
Read guide →Warfarin Pharmacokinetics Guide
Anticoagulation
Vitamin K antagonist
Read guide →Warfarin Pharmacokinetics Guide
Anticoagulation
Small Molecule
Read guide →Wegovy (Semaglutide) Pharmacokinetics Guide
Chronic weight management
GLP-1 RA
Read guide →Weight-HbA1c-Glucose Model Pharmacokinetics Guide
Obesity/T2DM
Small Molecule
Read guide →Xarelto (Rivaroxaban) Pharmacokinetics Guide
Stroke prevention in atrial fibrillation
Small Molecule
Read guide →Xolair (Omalizumab) Pharmacokinetics Guide
Moderate-to-severe allergic asthma
mAb
Read guide →Xtandi (Enzalutamide) Pharmacokinetics Guide
Metastatic castration-resistant prostate cancer
Small Molecule
Read guide →capecitabine Pharmacokinetics Guide
Fluoropyrimidine / Oral Prodrug
Read guide →evinacumab Pharmacokinetics Guide
HoFH
Monoclonal Antibody (ANGPTL3 Inhibitor)
Read guide →fda ruc Pharmacokinetics Guide
BRCA-mutated advanced ovarian, fallopian tube, or primary peritoneal cancer
PARP Inhibitor
Read guide →lenvatinib_Gupta_26879594 Pharmacokinetics Guide
Advanced renal cell carcinoma, hepatocellular carcinoma, differentiated thyroid cancer
Multikinase Inhibitor (TKI)
Read guide →mAb PBPK (Shah-Betts) Pharmacokinetics Guide
Monoclonal Antibodies
mAb
Read guide →mAb TMDD Platform Model Pharmacokinetics Guide
Monoclonal Antibodies
mAb
Read guide →mRNA-3927 Pharmacokinetics Guide
Propionic Acidemia
mRNA-LNP
Read guide →model replication (Benkali_et al) Pharmacokinetics Guide
Calcineurin Inhibitor
Read guide →poppk model of osimertinib Pharmacokinetics Guide
EGFR Tyrosine Kinase Inhibitor
Read guide →rucaparib ok model Pharmacokinetics Guide
Ovarian cancer, metastatic castration-resistant prostate cancer (mCRPC)
PARP Inhibitor
Read guide →rucaparib Pharmacokinetics Guide
BRCA-mutated advanced ovarian, fallopian tube, or primary peritoneal cancer
PARP Inhibitor
Read guide →semaglutide Pharmacokinetics Guide
Obesity (BMI ≥30) and overweight (BMI ≥27) with weight-related comorbidity; Type 2 Diabetes
GLP-1 Receptor Agonist
Read guide →siRNA Pharmacokinetics Guide
Various (gene silencing platform)
Small Interfering RNA (siRNA)
Read guide →test Pharmacokinetics Guide
Parasitic infections, immunomodulation (research)
Imidazothiazole (Immunomodulant/Anthelmintic)
Read guide →trastuzumab csf Pharmacokinetics Guide
HER2+ breast cancer with leptomeningeal metastases
Monoclonal Antibody (Anti-HER2)
Read guide →Build Your Own PK/PD Simulator
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